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{ "item_title" : "Functional Selectivity of G Protein-Coupled Receptor Ligands", "item_author" : [" Kim Neve "], "item_description" : "Historical Overview of the Concept of Functional Selectivity.- Functional Selectivity: Theoretical Considerations and Future Directions.- Agonist Selective Coupling of G Protein-Coupled Receptors.- Ligand-Selective Receptor Desensitization and Endocytosis.- Selectivity for G protein or Arrestin-Mediated Signaling.- In Vivo Evidence for and Consequences of Functional Selectivity.- Functional Selectivity at Adrenergic Receptors.- Signaling Diversity Mediated by Muscarinic Acetylcholine Receptor Subtypes and Evidence for Functional Selectivity.- Functional Selectivity at Serotonin Receptors.- Functional Selectivity at Dopamine Receptors.- Functional Selectivity at Receptors for Cannabinoids and other Lipids.- Functional Selectivity at Opioid Receptors Graciela Pi eyro.- Functional Selectivity at non-Opioid Peptide Receptors", "item_img_path" : "https://covers1.booksamillion.com/covers/bam/1/49/396/116/1493961160_b.jpg", "price_data" : { "retail_price" : "119.99", "online_price" : "119.99", "our_price" : "119.99", "club_price" : "119.99", "savings_pct" : "0", "savings_amt" : "0.00", "club_savings_pct" : "0", "club_savings_amt" : "0.00", "discount_pct" : "10", "store_price" : "" } }
Functional Selectivity of G Protein-Coupled Receptor Ligands|Kim Neve

Functional Selectivity of G Protein-Coupled Receptor Ligands : New Opportunities for Drug Discovery

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Overview

Historical Overview of the Concept of Functional Selectivity.- Functional Selectivity: Theoretical Considerations and Future Directions.- Agonist Selective Coupling of G Protein-Coupled Receptors.- Ligand-Selective Receptor Desensitization and Endocytosis.- Selectivity for G protein or Arrestin-Mediated Signaling.- In Vivo Evidence for and Consequences of Functional Selectivity.- Functional Selectivity at Adrenergic Receptors.- Signaling Diversity Mediated by Muscarinic Acetylcholine Receptor Subtypes and Evidence for Functional Selectivity.- Functional Selectivity at Serotonin Receptors.- Functional Selectivity at Dopamine Receptors.- Functional Selectivity at Receptors for Cannabinoids and other Lipids.- Functional Selectivity at Opioid Receptors Graciela Pi eyro.- Functional Selectivity at non-Opioid Peptide Receptors

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Details

  • ISBN-13: 9781493961160
  • ISBN-10: 1493961160
  • Publisher: Humana
  • Publish Date: August 2016
  • Dimensions: 9.21 x 6.14 x 0.64 inches
  • Shipping Weight: 0.94 pounds
  • Page Count: 292

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