Functional Selectivity of G Protein-Coupled Receptor Ligands : New Opportunities for Drug Discovery
Overview
Historical Overview of the Concept of Functional Selectivity.- Functional Selectivity: Theoretical Considerations and Future Directions.- Agonist Selective Coupling of G Protein-Coupled Receptors.- Ligand-Selective Receptor Desensitization and Endocytosis.- Selectivity for G protein or Arrestin-Mediated Signaling.- In Vivo Evidence for and Consequences of Functional Selectivity.- Functional Selectivity at Adrenergic Receptors.- Signaling Diversity Mediated by Muscarinic Acetylcholine Receptor Subtypes and Evidence for Functional Selectivity.- Functional Selectivity at Serotonin Receptors.- Functional Selectivity at Dopamine Receptors.- Functional Selectivity at Receptors for Cannabinoids and other Lipids.- Functional Selectivity at Opioid Receptors Graciela Pi eyro.- Functional Selectivity at non-Opioid Peptide Receptors
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Details
- ISBN-13: 9781493961160
- ISBN-10: 1493961160
- Publisher: Humana
- Publish Date: August 2016
- Dimensions: 9.21 x 6.14 x 0.64 inches
- Shipping Weight: 0.94 pounds
- Page Count: 292
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